Molecule Details
InChIKeySFNAMCXZMSYPAU-UHFFFAOYSA-N
Compound Name4-[[3-Piperidin-1-yl-1-[3-(pyridin-2-ylamino)phenyl]propyl]amino]quinazoline-8-carboxamide
Canonical SMILESNC(=O)c1cccc2c(NC(CCN3CCCCC3)c3cccc(Nc4ccccn4)c3)ncnc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.59
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 8.8 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 6.1 IC50 ChEMBL;BindingDB