Molecule Details
InChIKeySFHXUNXRQNJLAE-UHFFFAOYSA-N
Compound Name4-(4-Cyanoanilino)-6-piperazin-1-yl-1,3,5-triazine-2-carbonitrile
Canonical SMILESN#Cc1ccc(Nc2nc(C#N)nc(N3CCNCC3)n2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P43235 CTSK Homo sapiens Human PF08246 PF00112 7.5 IC50 ChEMBL;BindingDB
P07858 CTSB Homo sapiens Human PF00112 PF08127 7.2 IC50 ChEMBL;BindingDB
P07711 CTSL Homo sapiens Human PF08246 PF00112 7.0 IC50 ChEMBL;BindingDB