Molecule Details
InChIKeySEMWGSNVOBRKQC-QMMMGPOBSA-N
Compound Name3-(2-amino-1H-benzimidazol-4-yl)-6-[(2S)-2,3-diaminopropyl]sulfonyl-2-(2H-tetrazol-5-yl)benzenesulfonamide
Canonical SMILESNC[C@H](N)CS(=O)(=O)c1ccc(-c2cccc3[nH]c(N)nc23)c(-c2nnn[nH]2)c1S(N)(=O)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.34
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.8 IC50 ChEMBL;BindingDB
Q9XAY4 blaVIM Pseudomonas aeruginosa Pathogen PF00753 9.3 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 8.9 IC50 BindingDB