Molecule Details
InChIKeySDUVOQLCGBPUHH-UHFFFAOYSA-N
Compound NameAminoimidazo[1,2-a]pyridine deriv. 16
Canonical SMILESCOc1cc(F)c(C(=O)c2c(N)nc3ccc(C(=O)c4c(F)cccc4F)cn23)c(F)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.99
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P24941 CDK2 Homo sapiens Human PF00069 7.0 pIC50 TTD_MultiTarget
P06493 CDK1 Homo sapiens Human PF00069 7.0 pIC50 TTD_MultiTarget
P11802 CDK4 Homo sapiens Human PF00069 7.0 pIC50 TTD_MultiTarget