Molecule Details
InChIKeySDGJBAUIGHSMRI-UHFFFAOYSA-N
Compound NameN-(3-((5-Chloro-2-((2-methoxy-4-(4-methyl-1-piperazinyl)phenyl)amino)-4-pyrimidinyl)oxy)phenyl)propanamide
Canonical SMILESCCC(=O)Nc1cccc(Oc2nc(Nc3ccc(N4CCN(C)CC4)cc3OC)ncc2Cl)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.38
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O60285 NUAK1 Homo sapiens Human PF00069 8.3 IC50 ChEMBL;BindingDB
Q9H093 NUAK2 Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB
P00533 EGFR Homo sapiens Human PF00757 PF14843 PF07714 PF01030 PF21314 6.9 Kd ChEMBL