Molecule Details
InChIKeySDELPNZPQHTXIM-UHFFFAOYSA-N
Compound NameUS8835436, Example 134
Canonical SMILESCOc1ccc(-n2cc(C(=O)NCCCN3CCN(c4cccc(C)c4C)CC3)nc2-c2ccccc2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.36
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28223 HTR2A Homo sapiens Human PF00001 7.7 IC50 ChEMBL;BindingDB
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 7.4 IC50 ChEMBL;BindingDB
P28335 HTR2C Homo sapiens Human PF00001 7.0 IC50 ChEMBL;BindingDB