Molecule Details
InChIKeySDDRDZUPYOUOOW-UHFFFAOYSA-N
Compound Name2-[3-Biphenyl-2-ylmethyl-2-ethyl-8-(2-oxo-propoxy)-indolizin-1-yl]-2-oxo-acetamide
Canonical SMILESCCc1c(C(=O)C(N)=O)c2c(OCC(C)=O)cccn2c1Cc1ccccc1-c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.29
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P14555 PLA2G2A Homo sapiens Human PF00068 7.5 IC50 ChEMBL;BindingDB
Q9NZK7 PLA2G2E Homo sapiens Human PF00068 7.0 IC50 ChEMBL;BindingDB