Molecule Details
InChIKeySCUZVSHLJVHGDP-UHFFFAOYSA-N
Compound Name3-[[4-(2,6-dipyrrolidin-1-ylpyrimidin-4-yl)piperazin-1-yl]methyl]-2,5,7,8-tetramethyl-3,4-dihydro-2H-chromen-6-ol
Canonical SMILESCc1c(C)c2c(c(C)c1O)CC(CN1CCN(c3cc(N4CCCC4)nc(N4CCCC4)n3)CC1)C(C)O2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.82
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29466 CASP1 Homo sapiens Human PF00619 PF00656 7.3 Ki ChEMBL;BindingDB
P51878 CASP5 Homo sapiens Human PF00619 PF00656 6.8 IC50 ChEMBL;BindingDB
P49662 CASP4 Homo sapiens Human PF00619 PF00656 6.4 IC50 ChEMBL;BindingDB