Molecule Details
InChIKeySCHOOHHHHFRCGE-SMNOQFDKSA-N
Canonical SMILESCOC(=O)C12CCC(CC1)N(Cc1nc(C(F)(F)F)c(N[C@H]3CCc4c(-c5cccc(-c6ccc(CNC[C@@H]7CCC(=O)N7)c(OC)n6)c5Cl)cccc43)nc1OC)C2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL9.85
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15116 PDCD1 Homo sapiens Human PF07686 9.8 IC50 ChEMBL;BindingDB
Q9NZQ7 CD274 Homo sapiens Human PF08205 PF07686 9.8 IC50 ChEMBL