Molecule Details
InChIKeySCANZEHBHPIJEQ-CMDGGOBGSA-N
Compound NameN-(4-methyl-3-(3-((4-methylpiperazin-1-yl)methyl)styryl)-1H-indazol-5-yl)-2-(thiophen-2-yl)acetamide
Canonical SMILESCc1c(NC(=O)Cc2cccs2)ccc2[nH]nc(/C=C/c3cccc(CN4CCN(C)CC4)c3)c12
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.0
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O75716 STK16 Homo sapiens Human PF00069 7.0 pIC50 TTD_MultiTarget
Q96GD4 AURKB Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB