Molecule Details
InChIKeySBDOCCVDBJLSLR-JOCHJYFZSA-N
Compound NameUS9890166, Example 126
Canonical SMILESCOc1ccc(-c2nc3c([nH]2)[C@@H](c2ccc(Cl)cc2)N(c2cc(OC)c4nnc(C)n4c2)C3=O)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.65
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O60885 BRD4 Homo sapiens Human PF17035 PF17105 PF00439 7.0 IC50 ChEMBL;BindingDB
Q15059 BRD3 Homo sapiens Human PF17035 PF00439 6.5 IC50 ChEMBL;BindingDB
P25440 BRD2 Homo sapiens Human PF17035 PF00439 6.4 IC50 ChEMBL;BindingDB