Molecule Details
InChIKeySAXIOFYKEIRMET-ACZUPFTQSA-N
Canonical SMILESCC(=O)c1ccc(/C=C/CO[C@@H](C(=O)NNC(=O)CCc2ccccc2)[C@H](O)[C@@H](O)[C@@H](OC/C=C/c2ccc(C(C)=O)cc2)C(=O)N[C@H]2c3ccccc3C[C@H]2O)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.13
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P39898 PMI Plasmodium falciparum (isolate HB3) Pathogen PF00026 7.4 Ki ChEMBL;BindingDB
P46925 PMII Plasmodium falciparum (isolate HB3) Pathogen PF00026 6.8 Ki ChEMBL;BindingDB