Molecule Details
InChIKeySAOHYTLBHRCWIT-UHFFFAOYSA-N
Compound Name4-(1H-Imidazol-1-ylmethyl)-7-{[3-(trifluoromethoxy)benzyl]oxy}-2H-chromen-2-one
Canonical SMILESO=c1cc(Cn2ccnc2)c2ccc(OCc3cccc(OC(F)(F)F)c3)cc2o1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.29
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P15538 CYP11B1 Homo sapiens Human PF00067 8.3 IC50 ChEMBL;BindingDB
P19099 CYP11B2 Homo sapiens Human PF00067 6.9 IC50 ChEMBL;BindingDB
P11511 CYP19A1 Homo sapiens Human PF00067 6.7 IC50 ChEMBL;BindingDB