Molecule Details
InChIKeySAGGCAPQVJYEGE-UHFFFAOYSA-N
Compound NameN-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-2-(methylamino)-2-phenylacetamide
Canonical SMILESCNC(C(=O)Nc1cc2cc[nH]c(=O)c2cc1Cl)c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.58
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O75116 ROCK2 Homo sapiens Human PF25346 PF00069 PF08912 7.9 IC50 ChEMBL;BindingDB
Q13464 ROCK1 Homo sapiens Human PF25346 PF00069 PF08912 7.8 IC50 ChEMBL;BindingDB
Q16513 PKN2 Homo sapiens Human PF02185 PF00069 PF00433 7.0 IC50 ChEMBL;BindingDB