Target not found.
Molecule Details
InChIKeyRZSANBVXVBZRFN-UHFFFAOYSA-N
Compound Name4-[(3-chloro-N-pyrazin-2-ylanilino)methyl]-7,8-difluoro-1H-quinolin-2-one
Canonical SMILESO=c1cc(CN(c2cccc(Cl)c2)c2cnccn2)c2ccc(F)c(F)c2[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.11
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P35228 NOS2 Homo sapiens Human PF00667 PF00258 PF00175 PF02898 8.3 IC50 ChEMBL;BindingDB
P29475 NOS1 Homo sapiens Human PF00667 PF00258 PF00175 PF02898 PF00595 7.9 IC50 ChEMBL;BindingDB