Molecule Details
InChIKeyRZJPYZWXIJSYFQ-UHFFFAOYSA-N
Compound Name2-{4-[4-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-piperidin-1-yl]-butyl}-isoindole-1,3-dione
Canonical SMILESO=C1c2ccccc2C(=O)N1CCCCN1CCC(n2c(O)nc3ccccc32)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.62
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 9.6 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 8.5 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB