Molecule Details
InChIKeyRZJAOODRKRAJBF-UHFFFAOYSA-N
Canonical SMILESCc1cc(N2C(=O)c3nc(C4=CCN(C(=O)NC(C)(C)C)CC4)n(C(C)C)c3C2c2ccc(Cl)cc2)cn2c(C)nnc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.78
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O60885 BRD4 Homo sapiens Human PF17035 PF17105 PF00439 7.9 IC50 ChEMBL;BindingDB
P25440 BRD2 Homo sapiens Human PF17035 PF00439 7.6 IC50 ChEMBL;BindingDB