Molecule Details
InChIKeyRZBCPMYJIARMGV-UHFFFAOYSA-N
Canonical SMILESCOc1ncc(-c2ccc3c(Nc4cc(Oc5cc(F)cc(F)c5)cc(C(=O)O)c4)c(S(=O)(=O)NC4CC4)cnc3c2)c(OC)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.92
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P00338 LDHA Homo sapiens Human PF02866 PF00056 8.5 IC50 ChEMBL;BindingDB
P07195 LDHB Homo sapiens Human PF02866 PF00056 7.4 IC50 ChEMBL;BindingDB