Molecule Details
InChIKeyRYXUPKGYPPPMSC-UHFFFAOYSA-N
Compound NameN~6~-Methyl-N~6~-(3,4,5-Trifluorophenyl)pyrido[2,3-D]pyrimidine-2,4,6-Triamine
Canonical SMILESCN(c1cc(F)c(F)c(F)c1)c1cnc2nc(N)nc(N)c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.73
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P00374 DHFR Homo sapiens Human PF00186 6.8 IC50 ChEMBL;BindingDB
P16184 Pneumocystis carinii Pathogen PF00186 6.6 IC50 ChEMBL