Molecule Details
InChIKeyRYPURVOUHFFJCE-UHFFFAOYSA-N
Compound Name2-[1-(3-Methyl-benzyl)-piperidin-4-yl]-1-(2-methyl-2,3-dihydro-indol-1-yl)-ethanone
Canonical SMILESCc1cccc(CN2CCC(CC(=O)N3c4ccccc4CC3C)CC2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.54
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P21917 DRD4 Homo sapiens Human PF00001 8.3 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB