Molecule Details
InChIKeyRYNRWNJFDSYFLB-TUCRWICHSA-N
Compound NameBoc-Trp-Phg-Asp-1Nal-NH2
Canonical SMILESCC(C)(C)OC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](Cc1cccc2ccccc12)C(N)=O)c1ccccc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.85
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32238 CCKAR Homo sapiens Human PF00001 PF09193 7.8 pIC50 TTD_MultiTarget
P32239 CCKBR Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB