Molecule Details
InChIKeyRYJMJCJWMWMLJV-UHFFFAOYSA-N
Compound NameN-cyclopropyl-2-[3-[4-[4-(1H-pyrazol-4-yl)anilino]-5,7-dihydrofuro[3,4-d]pyrimidin-2-yl]phenoxy]acetamide
Canonical SMILESO=C(COc1cccc(-c2nc3c(c(Nc4ccc(-c5cn[nH]c5)cc4)n2)COC3)c1)NC1CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.41
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11169 SLC2A3 Homo sapiens Human PF00083 6.6 IC50 ChEMBL;BindingDB
P11166 SLC2A1 Homo sapiens Human PF00083 6.2 IC50 ChEMBL;BindingDB
O97467 ht1 Plasmodium falciparum Pathogen PF00083 6.4 IC50 ChEMBL;BindingDB