Molecule Details
InChIKeyRYFBXXBUFPDLOZ-LLVKDONJSA-N
Compound Name2-amino-N-(2-aminoethyl)-5-chloro-3-[4-[[(3R)-pyrrolidin-3-yl]sulfamoyl]-3-sulfamoyl-2-(2H-tetrazol-5-yl)phenyl]benzamide
Canonical SMILESNCCNC(=O)c1cc(Cl)cc(-c2ccc(S(=O)(=O)N[C@@H]3CCNC3)c(S(N)(=O)=O)c2-c2nn[nH]n2)c1N
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL9.1
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q2QC95 blaoxa-10 Klebsiella pneumoniae Pathogen PF00905 9.6 IC50 BindingDB
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.3 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 8.5 IC50 BindingDB