Molecule Details
InChIKeyRXLCWZMWTUZMFM-UHFFFAOYSA-N
Compound Name7,8-dichloro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine
Canonical SMILESCN(C)C1(CNCCC2CCOCC2)COc2cc(Cl)c(Cl)cc2OC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.44
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08172 CHRM2 Homo sapiens Human PF00001 9.9 Ki ChEMBL;BindingDB
P20309 CHRM3 Homo sapiens Human PF00001 9.7 Ki ChEMBL;BindingDB
P11229 CHRM1 Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB