Molecule Details
InChIKeyRXDFGEFKYADZNK-UHFFFAOYSA-N
Compound Name3-Amino-N-[4-[4-(3-amino-1-oxopropyl)-1-piperazinyl]-3-pyridinyl]-2-pyrazinecarboxamide
Canonical SMILESNCCC(=O)N1CCN(c2ccncc2NC(=O)c2nccnc2N)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.72
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 7.2 Ki ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 6.7 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.2 Ki ChEMBL;BindingDB