Molecule Details
InChIKeyRVRPAIWBGBVSKB-UHFFFAOYSA-N
Compound Name1-[4-[[4-(4,5-dihydro-1H-imidazol-2-ylamino)phenyl]methyl]phenyl]-2-(furan-2-ylmethyl)guanidine
Canonical SMILESN=C(NCc1ccco1)Nc1ccc(Cc2ccc(NC3=NCCN3)cc2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.75
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08913 ADRA2A Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P18089 ADRA2B Homo sapiens Human PF00001 8.8 Ki ChEMBL
P18825 ADRA2C Homo sapiens Human PF00001 8.8 Ki ChEMBL