Molecule Details
InChIKeyRVPVTOKNUYGICG-UHFFFAOYSA-N
Compound NameN-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-(3-methoxyphenyl)picolinamide
Canonical SMILESCOc1cccc(-c2nc(C(=O)NCc3ccc([S@SP2](C)(=O)=O)cc3)cc(N)c2C#N)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.29
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 6.4 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB