Molecule Details
InChIKeyRVCUOIJKDXETPG-UHFFFAOYSA-N
Compound Name3-(2,3,3a,4,6,6a-hexahydro-1H-pyrrolo[3,4-c]pyrrol-5-yl)-1-(1-cyclooctylpiperidin-4-yl)pyrido[2,3-b]pyrazin-2-one
Canonical SMILESO=c1c(N2CC3CNCC3C2)nc2ncccc2n1C1CCN(C2CCCCCCC2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.96
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5TC84 OGFRL1 Homo sapiens Human PF04664 7.3 Ki ChEMBL;BindingDB
P41145 OPRK1 Homo sapiens Human PF00001 6.9 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB