Molecule Details
InChIKeyRVBIHRGXDKNPKO-UHFFFAOYSA-N
Compound Name2-(1,3-dioxoisoindolin-2-yl)-N-(4-sulfamoylphenethyl)acetamide
Canonical SMILESNS(=O)(=O)c1ccc(CCNC(=O)CN2C(=O)c3ccccc3C2=O)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.3
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16790 CA9 Homo sapiens Human PF00194 6.5 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 6.2 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 6.2 pIC50 TTD_MultiTarget