Molecule Details
InChIKeyRVBDWZKWSXQLMF-DOTOQJQBSA-N
Compound NameN-((3R,4R)-1-Benzyl-4-methyl-pyrrolidin-3-ylmethyl)-5-chloro-2-methoxy-4-methylamino-benzamide
Canonical SMILESCNc1cc(OC)c(C(=O)NC[C@@H]2CN(Cc3ccccc3)C[C@@H]2C)cc1Cl
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.78
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14416 DRD2 Homo sapiens Human PF00001 7.5 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB