Molecule Details
InChIKeyRUQVXLIOJPKNCM-JTQLQIEISA-N
Compound Name6-methyl-5-[(3R)-3-(3,4,5-trimethoxyphenyl)but-1-ynyl]pyrimidine-2,4-diamine
Canonical SMILESCOc1cc([C@@H](C)C#Cc2c(C)nc(N)nc2N)cc(OC)c1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.64
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q07422 Toxoplasma gondii Pathogen PF00186 PF00303 8.8 IC50 ChEMBL;BindingDB
Q27552 DHFR-TS Cryptosporidium parvum Pathogen PF00186 PF00303 7.1 IC50 ChEMBL;BindingDB
P22906 DFR1 Candida albicans Pathogen PF00186 7.0 IC50 ChEMBL;BindingDB