Molecule Details
InChIKeyRUJOXQDERXMGDN-UHFFFAOYSA-N
Compound Name2-(5-Chloro-2-hydroxy-biphenyl-3-yl)-1H-benzoimidazole-5-carboxamidine
Canonical SMILESN=C(N)c1ccc2[nH]c(-c3cc(Cl)cc(-c4ccccc4)c3O)nc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.29
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00750 PLAT Homo sapiens Human PF00008 PF00039 PF00051 PF00089 6.5 Ki ChEMBL;BindingDB
P00749 PLAU Homo sapiens Human PF00051 PF00089 6.3 Ki ChEMBL;BindingDB
P00742 F10 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 6.0 Ki ChEMBL;BindingDB