Molecule Details
InChIKeyRUGBLRYISYKONW-UHFFFAOYSA-N
Compound NameN-(2-methoxy-6-methyl-1-prop-2-ynoxy-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)butanamide
Canonical SMILESC#CCOc1c(OC)cc2c3c1-c1cc(NC(=O)CCC)ccc1CC3N(C)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.32
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P50406 HTR6 Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB
P34969 HTR7 Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB