Molecule Details
InChIKeyRUCWXMRMXGLFKN-UHFFFAOYSA-N
Compound Name1-(4-Amino-5-chloro-2-methoxyphenyl)-3-[1-[(piperidin-4-yl)methyl]-4-piperidyl] propan-1-one
Canonical SMILESCOc1cc(N)c(Cl)cc1C(=O)CCC1CCN(CC2CCNCC2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.76
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13639 HTR4 Homo sapiens Human PF00001 8.6 Ki ChEMBL;BindingDB
P22303 ACHE Homo sapiens Human PF08674 PF00135 6.9 IC50 ChEMBL;BindingDB