Molecule Details
InChIKeyRTPDDFLFZXREMW-BQYQJAHWSA-N
Compound Name8-(Pyrimidin-2-ylamino)-6-((E)-styryl)-naphthalene-2-carboxamidine
Canonical SMILESN=C(N)c1ccc2cc(/C=C/c3ccccc3)cc(Nc3ncccn3)c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.31
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00749 PLAU Homo sapiens Human PF00051 PF00089 8.0 Ki ChEMBL;BindingDB
P06870 KLK1 Homo sapiens Human PF00089 7.4 Ki ChEMBL;BindingDB
P00747 PLG Homo sapiens Human PF00051 PF00024 PF00089 6.6 Ki ChEMBL;BindingDB