Molecule Details
InChIKeyRTHKPHCVZVYDFN-UHFFFAOYSA-N
Canonical SMILESNc1nccc(-c2c3c(O)ccnc3n3c(N)nccc23)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.34
SourceChEMBL
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB08694
Drug NameVariolin B
CAS Numbernan
Groups experimental
ATC Codes nan
Descriptionnan

Categories: Alkaloids
Cross-references: BindingDB: 50398327 CHEMBL380500 ChemSpider: 7993300 PDB: VAR PubChem:9817550 PubChem:99445165 ZINC: ZINC000020149024
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P50750 CDK9 Homo sapiens Human PF00069 7.6 IC50 ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 7.1 IC50 ChEMBL
DrugBank Target Actions (2)
Target Gene Target Name Action Type
P20248 CCNA2 Cyclin-A2 binder targets
P24941 CDK2 Cyclin-dependent kinase 2 binder targets