Molecule Details
InChIKeyRTFQFPZKDYMMMJ-RIAKQDHQSA-N
Canonical SMILESCc1ccc(F)c(S(=O)(=O)Nc2ccc(-c3nc(OC[C@H]4CN(CCCCCCOCCOCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)CCO4)c4cn[nH]c4n3)cc2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.59
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O00141 SGK1 Homo sapiens Human PF00069 PF00433 6.7 IC50 ChEMBL
Q96BR1 SGK3 Homo sapiens Human PF00069 PF00433 PF00787 6.5 IC50 ChEMBL