Molecule Details
InChIKeyRSSMYFQRFUEXTN-JKDDQTOVSA-N
Canonical SMILESC[C@@](NCc1ccc2ncsc2c1)(c1cn(C(CCS(C)(=O)=O)C(=O)COc2c(F)c(F)cc(F)c2F)nn1)C1CCCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.15
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P08684 CYP3A4 Homo sapiens Human PF00067 6.7 IC50 ChEMBL;BindingDB
P25779 Trypanosoma cruzi Pathogen PF12131 PF08246 PF00112 7.6 IC50 ChEMBL;BindingDB