Molecule Details
InChIKeyRRZKRPHYMGDLBB-ZZHFZYNASA-N
Compound Name{1-[5-(2-Fluoro-phenyl)-1-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-ylcarbamoyl]-2-phenyl-ethyl}-carbamic acid tert-butyl ester
Canonical SMILESCN1C(=O)C(NC(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)N=C(c2ccccc2F)c2ccccc21
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.0
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32238 CCKAR Homo sapiens Human PF00001 PF09193 6.0 pIC50 TTD_MultiTarget
P32239 CCKBR Homo sapiens Human PF00001 6.0 IC50 ChEMBL