Molecule Details
InChIKeyRRWISUYOSRHAFZ-QYBDOPJKSA-N
Compound Name(S)-1-(2-((S)-4-(6-fluoronaphthalen-2-yl)-2-methylpiperazin-1-yl)ethyl)isochroman-6-carboxamide
Canonical SMILESC[C@H]1CN(c2ccc3cc(F)ccc3c2)CCN1CC[C@@H]1OCCc2cc(C(N)=O)ccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.68
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 8.7 Ki ChEMBL;BindingDB
P28221 HTR1D Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB