Molecule Details
InChIKeyRROPCZKHYUPTGO-UHFFFAOYSA-N
Compound Name2-(7-(2-Methoxyethoxy)imidazo[1,2-a]pyridin-3-yl)-8-(piperidin-4-yloxy)quinoline
Canonical SMILESCOCCOc1ccn2c(-c3ccc4cccc(OC5CCNCC5)c4n3)cnc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.38
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 8.7 IC50 ChEMBL;BindingDB
P35968 KDR Homo sapiens Human PF07679 PF00047 PF13895 PF22971 PF07714 PF21339 PF17988 PF22854 7.4 IC50 ChEMBL
P10721 KIT Homo sapiens Human PF00047 PF07714 6.0 IC50 ChEMBL