Molecule Details
InChIKeyRRLCBKCJYXFQHA-UHFFFAOYSA-N
Compound Name2-[4-(3-Thiophen-3-yl-benzyl)-piperazin-1-yl]-pyrimidine
Canonical SMILESc1cnc(N2CCN(Cc3cccc(-c4ccsc4)c3)CC2)nc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21917 DRD4 Homo sapiens Human PF00001 8.5 IC50 ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 6.7 IC50 ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.5 IC50 ChEMBL;BindingDB