Molecule Details
InChIKeyRRHZICZHWYWVEE-UHFFFAOYSA-N
Compound Name4-(6-(5-(1,3,4-thiadiazol-2-yl)-1H-indol-3-yl)pyridin-2-yl)morpholine
Canonical SMILESc1cc(-c2c[nH]c3ccc(-c4nncs4)cc23)nc(N2CCOCC2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB