Molecule Details
InChIKeyRREWXFWIJFLGBI-UHFFFAOYSA-N
Compound Name6-(aminomethyl)-5-(2,4-dichlorophenyl)-N-(1-ethyl-1H-pyrazol-5-yl)-7-methylimidazo(1,2-a)pyrimidine-2-carboxamide
Canonical SMILESCCn1nccc1NC(=O)c1cn2c(-c3ccc(Cl)cc3Cl)c(CN)c(C)nc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.97
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86TI2 DPP9 Homo sapiens Human PF19520 PF00930 PF00326 9.1 Ki ChEMBL;BindingDB
P27487 DPP4 Homo sapiens Human PF00930 PF00326 9.0 Ki ChEMBL;BindingDB
Q6V1X1 DPP8 Homo sapiens Human PF19520 PF00930 PF00326 8.9 Ki ChEMBL;BindingDB