Molecule Details
InChIKeyRQZHKEFEFWSLOK-PHNIDTBTSA-N
Compound NameAc-Arg-Cys-D-Ala-His-D-Phe-Arg-Trp-Cys-NH2
Canonical SMILESCC(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CS)C(=O)N[C@H](C)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@H](Cc1ccccc1)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CS)C(N)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.23
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q01726 MC1R Homo sapiens Human PF00001 8.5 Ki ChEMBL;BindingDB
P32245 MC4R Homo sapiens Human PF00001 8.4 Ki ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB