Molecule Details
InChIKeyRQYMSPDZFNAIFN-CYBMUJFWSA-N
Compound Name5-[3-[6-[(3R)-3-methylpiperidin-1-yl]-2-pyridinyl]-1H-indol-5-yl]-1,3,4-thiadiazol-2-amine
Canonical SMILESC[C@@H]1CCCN(c2cccc(-c3c[nH]c4ccc(-c5nnc(N)s5)cc34)n2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.27
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB