Molecule Details
InChIKeyRQUGSKZRACGFFU-UHFFFAOYSA-N
Compound NameN-(4-(3-morpholino-1H-1,2,4-triazol-1-yl)phenyl)-8-(thiazol-2-yl)quinazolin-2-amine
Canonical SMILESc1cc(-c2nccs2)c2nc(Nc3ccc(-n4cnc(N5CCOCC5)n4)cc3)ncc2c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.83
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P53779 MAPK10 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB