Molecule Details
InChIKeyRQQPWZPNFCJSRC-UHFFFAOYSA-N
Compound Name4-[2-(2-Fluoro-5-methylanilino)pyrimidin-4-yl]benzenesulfonamide
Canonical SMILESCc1ccc(F)c(Nc2nccc(-c3ccc(S(N)(=O)=O)cc3)n2)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.5
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P24941 CDK2 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
P11802 CDK4 Homo sapiens Human PF00069 7.5 pIC50 TTD_MultiTarget