Molecule Details
InChIKeyRQNOIZBVICJIJP-UHFFFAOYSA-N
Compound NameN-[5-(2-methoxyphenoxy)-2-morpholin-4-yl-6-[2-(propylsulfonylamino)ethoxy]pyrimidin-4-yl]-5-propan-2-ylpyridine-2-sulfonamide
Canonical SMILESCCCS(=O)(=O)NCCOc1nc(N2CCOCC2)nc(NS(=O)(=O)c2ccc(C(C)C)cn2)c1Oc1ccccc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.92
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P24530 EDNRB Homo sapiens Human PF00001 7.0 IC50 ChEMBL;BindingDB
P25101 EDNRA Homo sapiens Human PF00001 6.8 IC50 ChEMBL;BindingDB