Molecule Details
InChIKeyRQFQNQBNKTWWPR-UHFFFAOYSA-N
Compound Name2-cyano-4-(cyclohexylmethoxy)-N-phenethylpyrimidine-5-carboxamide
Canonical SMILESN#Cc1ncc(C(=O)NCCc2ccccc2)c(OCC2CCCCC2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.34
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P43235 CTSK Homo sapiens Human PF08246 PF00112 8.1 IC50 ChEMBL;BindingDB
P25774 CTSS Homo sapiens Human PF08246 PF00112 7.8 IC50 ChEMBL;BindingDB
P07711 CTSL Homo sapiens Human PF08246 PF00112 6.1 IC50 ChEMBL;BindingDB